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ヘテロサイクルの指向されたC-H機能化の限界を克服する

Yue-Jin Liu1, Hui Xu1, Wei-Jun Kong1

  • 1State Key Laboratory of Organometallic Chemistry, Shanghai Institute of Organic Chemistry, Chinese Academy of Sciences, 345 Lingling Road, Shanghai 200032, China.

Nature
|November 11, 2014
PubMed
まとめ

この研究は,ヘテロサイクルのC-H活性化を誘導する新しい方法を導入し,窒素と硫黄原子による触媒毒を克服します. N-メトキシアミド群は選択的機能化を可能にし,薬剤発見のアプリケーションを進める.

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