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Updated: Mar 29, 2026

Protocol for the Synthesis of Ortho-trifluoromethoxylated Aniline Derivatives
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Published on: January 19, 2016

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α-およびβ-フッ化アミドの直接触媒非対称マニッヒ型反応

Lennart Brewitz, Fernando Arteaga Arteaga, Liang Yin1

  • 1Institute of Microbial Chemistry (BIKAKEN) , Tokyo, Kamiosaki 3-14-23, Shinagawa-ku, Tokyo 141-0021, Japan.

Journal of the American Chemical Society
|December 15, 2015
PubMed
まとめ

直接エノライゼーションは,新しい触媒システムを用いて,フッ素アミノ酸を効率的に合成します. この方法により,薬剤化学のための価値あるキラル構成要素へのアクセスを可能にします.

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