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Updated: Mar 28, 2026

Preparation of N-2-alkoxyvinylsulfonamides from N-tosyl-1,2,3-triazoles and Subsequent Conversion to Substituted Phthalans and Phenethylamines
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Preparation of N-2-alkoxyvinylsulfonamides from N-tosyl-1,2,3-triazoles and Subsequent Conversion to Substituted Phthalans and Phenethylamines

Published on: January 3, 2018

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N-クロロアミドを用いたサイト選択C-H塩化により,クロロリスオクリミドの合成が可能

Ryan K Quinn1, Zef A Könst2, Sharon E Michalak2

  • 1Department of Chemistry, The University of North Carolina at Chapel Hill , Chapel Hill, North Carolina 27599, United States.

Journal of the American Chemical Society
|December 24, 2015
PubMed
まとめ

この研究は,N-クロロアミドを用いてアリファティックC-H結合を塩素化するための選択的方法を導入する. クロロリスオクリミドのような 複雑な分子の効率的な合成を可能にします 潜在的な癌治療薬です

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