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Updated: Mar 17, 2026

Preparation of Enantiopure Non-Activated Aziridines and Synthesis of Biemamide B, D, and epiallo-Isomuscarine
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エナチオセレクティブ・トータル・シンセシス (+) - プシグアディアルB

Lauren M Chapman1, Jordan C Beck1, Linglin Wu1

  • 1The Warren and Katharine Schlinger Laboratory for Chemistry and Chemical Engineering, Division of Chemistry and Chemical Engineering, California Institute of Technology , Pasadena, California 91125, United States.

Journal of the American Chemical Society
|July 26, 2016
PubMed
まとめ

この研究は,細胞毒性のある天然産物である (+) - サイグアディアルBの最初の全合成を報告した. 主なステップは,非対称なケテン添加,C ((sp3) -Hアルケニル化,およびテルペンフレーム構造のための環閉メタテシスであった.

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