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Updated: Mar 15, 2026

Amide Coupling Reaction for the Synthesis of Bispyridine-based Ligands and Their Complexation to Platinum as Dinuclear Anticancer Agents
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Amide Coupling Reaction for the Synthesis of Bispyridine-based Ligands and Their Complexation to Platinum as Dinuclear Anticancer Agents

Published on: May 28, 2014

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ダイナミック・キネティック・アシンメトリック・ブッチャウォルド・ハートウィッグ・アミネーションによるIAN型N,N-リガンドの合成

Pedro Ramírez-López1, Abel Ros1,2, Antonio Romero-Arenas1

  • 1Instituto Investigaciones Químicas (CSIC-US) , C/Américo Vespucio, 49, 41092 Sevilla, Spain.

Journal of the American Chemical Society
|September 6, 2016
PubMed
まとめ

この研究は,パラジウム触媒とQUINAPリガンドを使用してキラルアミンを生成する新しい方法を導入しています. このプロセスは高収量とエナチオ選択性を達成し,非対称合成のための貴重なツールを提供します.

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