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Updated: Mar 6, 2026

Preparation of Enantiopure Non-Activated Aziridines and Synthesis of Biemamide B, D, and epiallo-Isomuscarine
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Preparation of Enantiopure Non-Activated Aziridines and Synthesis of Biemamide B, D, and epiallo-Isomuscarine

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アントロンの非対称性アルキル化, (-) -および (+) -ヴィリジカトトキシンBおよびその同類物のエナンチオセレクティブ・トータル・シンセシス:絶対構成および強力な抗菌剤

K C Nicolaou1, Guodu Liu1, Kathryn Beabout1

  • 1Department of Chemistry, BioScience Research Collaborative and ‡Department of Biochemistry and Cell Biology, Rice University , 6100 Main Street, Houston, Texas 77005, United States.

Journal of the American Chemical Society
|March 4, 2017
PubMed
まとめ

新しい非対称性アルキル化法により,エナチオピュアなビリジカトキシンBおよび関連類の効率的な合成が可能である. この非対称合成の突破は 新しい抗菌剤の発見を容易にするでしょう

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