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Updated: Mar 1, 2026

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ペプチドアゴニストと結合するGLP-1受容体の結晶構造

Ali Jazayeri1, Mathieu Rappas1, Alastair J H Brown1

  • 1Heptares Therapeutics Ltd, BioPark, Broadwater Road, Welwyn Garden City, Hertfordshire AL7 3AX, UK.

Nature
|June 1, 2017
PubMed
まとめ

研究者は,ペプチドアゴニストと結合するグルカゴン型ペプチド1 (GLP- 1) 受容体の結晶構造を決定した. この構造的な洞察は,糖尿病の治療に強力な活性を持つ新しいペプチドアゴニストの設計を導いた.

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