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Updated: Feb 27, 2026

Author Spotlight: Evaluating Biophysical Assays for Characterizing PROTACS Ternary Complexes
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Author Spotlight: Evaluating Biophysical Assays for Characterizing PROTACS Ternary Complexes

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K2P2.1 (TREK-1) -アクティベーター複合体は,神秘的な選択性フィルター結合部位を明らかにする

Marco Lolicato1, Cristina Arrigoni1, Takahiro Mori2

  • 1Cardiovascular Research Institute, University of California, San Francisco, California 941158-9001, USA.

Nature
|July 11, 2017
PubMed
まとめ

研究者らは,TREK チャンネルを安定させることで活性化する小さな分子を発見しました.

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