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Updated: Feb 23, 2026

Synthesis of a Borylated Ibuprofen Derivative Through Suzuki Cross-Coupling and Alkene Boracarboxylation Reactions
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塩基に敏感なボロン酸による"カチオン"スズキ-ミヤウラ結合

Liye Chen1, Daniel R Sanchez1, Bufan Zhang1

  • 1Department of Chemistry, Princeton University , Princeton, New Jersey 08544, United States.

Journal of the American Chemical Society
|September 2, 2017
PubMed
まとめ

この研究では,新しい塩基なしのスズキ-ミヤウラ結合 (SMC) 方法が導入されています. この進歩により,過敏なポリフルオアリル化合物を含め,温和な条件下で効率的な結合が可能になります.

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