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Updated: Jan 26, 2026

Pharmacophore Modeling for Targets with Extensive Ligand Libraries: A Case Study on SARS-CoV-2 Mpro
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アルセノプラチン-1は,ダブル・ファルマコフォア抗がん剤である

Đenana Miodragović1,2, Antonello Merlino3, Elden P Swindell1

  • 1Chemistry of Life Processes Institute , Northwestern University , 2145 Sheridan Road , Evanston , Illinois 60208 , United States.

Journal of the American Chemical Society
|April 4, 2019
PubMed
まとめ

新しい抗がん剤であるアルセノプラチン-1は,その原薬と比較して,様々ながん細胞系に対する優れた活性を示しています. この化合物は プラチナとヒ素の両方を 癌細胞に効果的に送って 固体腫瘍を治療する可能性を秘めています

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