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Updated: Jan 3, 2026

Preparation of Enantiopure Non-Activated Aziridines and Synthesis of Biemamide B, D, and epiallo-Isomuscarine
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Preparation of Enantiopure Non-Activated Aziridines and Synthesis of Biemamide B, D, and epiallo-Isomuscarine

Published on: June 13, 2022

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アリファティックアミンのN-H結合に高度なエナンチオセレクティブカルベンの挿入

Mao-Lin Li1, Jin-Han Yu1, Yi-Hao Li1

  • 1State Key Laboratory and Institute of Elemento-Organic Chemistry, College of Chemistry, Nankai University, Tianjin 300071, China.

Science (New York, N.Y.)
|November 23, 2019
PubMed
まとめ

この研究では,アリファティックなアミンN-H結合にエナチオ選択カルベンの挿入のための新しいタンデム触媒法が導入されています. この革新的なアプローチは,触媒阻害を克服し,キラルアルファアミノ酸誘導体の合成を可能にします.

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