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(-) バクトボリンAのステレオ制御合成

Petra Vojáčková1,2, Lucyna Michalska1,2, Marek Nečas1

  • 1Department of Chemistry, Masaryk University, Brno 625 00, Czech Republic.

Journal of the American Chemical Society
|April 15, 2020
PubMed
まとめ

この研究では,抗腫瘍抗生物質 (-) - バクトボリンAのステレオ選択的合成が報告されています. この新しい経路では, (-) - キニン酸とキー反応を用いて分子を構成し,標的化合物の90 mgが得られます.

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