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Updated: Dec 22, 2025

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Pd-Catalyzed γ-C ((sp3) -H フリーアミンのフッ化

Yan-Qiao Chen1, Sukriti Singh2, Yongwei Wu1

  • 1Department of Chemistry, The Scripps Research Institute, 10550 N. Torrey Pines Road, La Jolla, California 92037, United States.

Journal of the American Chemical Society
|May 5, 2020
PubMed
まとめ

この研究は,新しい一時的誘導基を用いた自由アミンの最初の直接の γ-C ((sp3) -H 化を導入する. この方法は,メチルとメチレン位置でのアリファティックアミンを選択的にフッ素化し,新しい合成経路を提供します.

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