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Microwave-Assisted Preparation of 1-Aryl-1H-pyrazole-5-amines
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溶性弱塩基を用いたアリルアミネーション

Sii Hong Lau1, Peng Yu1, Liye Chen1

  • 1Department of Chemistry, Princeton University, Princeton, New Jersey 08544, United States.

Journal of the American Chemical Society
|November 12, 2020
PubMed
まとめ

この研究は,弱塩基としてトライエチラミン (Et3N) を使用した新しいパラジアム触媒C-N結合反応を導入します. この方法は,繊細な機能群に対応し,新しい合成戦略を可能にすることで,アミナ化反応の範囲を広げます.

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