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Cercosporin-Photocatalyzed [4+1]- and [4+2]-Annulations of Azoalkenes Under Mild Conditions
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制御されたN-サイト選択性を持つベンジルC-H結合とアゾールの銅触媒クロスカップリング

Si-Jie Chen1, Dung L Golden1, Shane W Krska2

  • 1Department of Chemistry, University of Wisconsin-Madison, 1101 University Avenue, Madison, Wisconsin 53706, United States.

Journal of the American Chemical Society
|August 31, 2021
PubMed
まとめ

この研究は,アゾールの部位選択的なN-H/C-Hクロスカップリングのための新しい銅触媒方法を示しています. このアプローチは選択性の課題を克服し,薬剤発見のための複雑な分子の効率的な合成を可能にします.

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