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Updated: Oct 1, 2025

Constructing Cyclic Peptides Using an On-Tether Sulfonium Center
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金 ((I) - プロパルギル化ペプチドのイミン形成による急速な循環

Rajeshwer Vanjari1, Deepanjan Panda1, Shaswati Mandal1

  • 1Schulich Faculty of Chemistry, Technion - Israel Institute of Technology, Haifa 3200008, Israel.

Journal of the American Chemical Society
|March 8, 2022
PubMed
まとめ

研究者たちは,保護されていないサイドチェーンの場合でも,様々な周期性ペプチドを合成するための迅速な金触媒方法を開発しました. このアプローチは効率的な薬剤発見と 治療の可能性のある新しい循環性ペプチドの作成を可能にします

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