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Updated: Sep 27, 2025

Facile Preparation of 2Z,4E-Dienamides by the Olefination of Electron-deficient Alkenes with Allyl Acetate
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アリルC−Hアミネーションクロスカップリングは,電離金属触媒によって三次アミンを供給する

Siraj Z Ali1, Brenna G Budaitis1, Devon F A Fontaine1

  • 1Roger Adams Laboratory, Department of Chemistry, University of Illinois, Urbana, IL 61801, USA.

Science (New York, N.Y.)
|April 14, 2022
PubMed
まとめ

研究者らは,薬剤で重要な複雑な三次アミンを合成するための新しいパラジウム触媒方法を開発しました. このアプローチはアミンによる触媒阻害を克服し,効率的なクロスカップリング反応を可能にします.

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