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Updated: Sep 24, 2025

Synthesis of a Borylated Ibuprofen Derivative Through Suzuki Cross-Coupling and Alkene Boracarboxylation Reactions
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Published on: November 30, 2022

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バスティモリドBのステレオ制御トータル合成は,ボロンエステルのイテラティブホモロゲーションを使用する

Daniele Fiorito1, Selbi Keskin1, Joseph M Bateman1

  • 1School of Chemistry, University of Bristol, Cantock's Close, Bristol BS8 1TS, U.K.

Journal of the American Chemical Society
|May 2, 2022
PubMed
まとめ

研究者たちは,抗マラリア剤 バスティモリドB の複雑な構造である 1,5-ポリオルを合成するための新しい方法を開発しました. この新しいアプローチにより 精密なステレオ制御が可能になり 複雑な分子の合成が容易になります

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