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Updated: Sep 22, 2025

Efficient Construction of Drug-like Bispirocyclic Scaffolds Via Organocatalytic Cycloadditions of α-Imino γ-Lactones and Alkylidene Pyrazolones
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Efficient Construction of Drug-like Bispirocyclic Scaffolds Via Organocatalytic Cycloadditions of α-Imino γ-Lactones and Alkylidene Pyrazolones

Published on: February 7, 2019

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ディカルボキシル酸のサイトセレクティブメチレンC-H乳酸化

Hau Sun Sam Chan1, Ji-Min Yang1, Jin-Quan Yu1

  • 1Department of Chemistry, The Scripps Research Institute, 10550 North Torrey Pines Road, La Jolla, CA 92037, USA.

Science (New York, N.Y.)
|May 26, 2022
PubMed
まとめ

研究者は,カルボキシル酸における選択的C−H結合活性化のための新しいパラジウム触媒方法を開発した. これは天然製品のような複雑な分子を作るのに有用な様々なラクトンの効率的な合成を可能にします.

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