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Updated: Sep 1, 2025

Detecting the Ligand-binding Domain Dimerization Activity of Estrogen Receptor Alpha Using the Mammalian Two-Hybrid Assay
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光スイッチ可能なディアゾシン基エストロゲン受容体アゴニスト:受容体内の活性形態の安定化

Julia Ewert1, Linda Heintze2, Mireia Jordà-Redondo3

  • 1Otto-Diels-Institute of Organic Chemistry, Christian-Albrechts-University of Kiel, 24098 Kiel, Germany.

Journal of the American Chemical Society
|August 11, 2022
PubMed
まとめ

この研究では 紫光で活性化し 緑色で無効化する 新種の光スイッチ薬が導入されました これらの化合物は高い標的特異性を示し,副作用と環境への影響を最小限に抑えています.

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