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Preparation of Enantiopure Non-Activated Aziridines and Synthesis of Biemamide B, D, and epiallo-Isomuscarine
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Preparation of Enantiopure Non-Activated Aziridines and Synthesis of Biemamide B, D, and epiallo-Isomuscarine

Published on: June 13, 2022

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(+) アベラロンの総合合成

Yang Wang1, Yongjian Su1, Yanxing Jia1

  • 1State Key Laboratory of Natural and Biomimetic Drugs, School of Pharmaceutical Sciences, and Chemical Biology Center, Peking University, 38 Xueyuan Road, Beijing 100191, China.

Journal of the American Chemical Society
|April 21, 2023
PubMed
まとめ

研究者は12段階で複合的なディテルペン (+) - アベラーロンを効率的に合成しました. トリキナンのこの新しい合成は,重要な非対称な触媒とラジカルカスケード反応を利用して,保護グループを回避します.

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