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Updated: Jul 27, 2025

Construction of Cyclic Cell-Penetrating Peptides for Enhanced Penetration of Biological Barriers
10:12

Construction of Cyclic Cell-Penetrating Peptides for Enhanced Penetration of Biological Barriers

Published on: September 19, 2022

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脂質膜を横断するペプチド輸送を制御する光スイッチ可能なカリキセレンアクティベーター

Joana N Martins1, Beatriz Raimundo1, Alicia Rioboo2

  • 1Laboratório Associado para a Química Verde (LAQV), Rede de Química e Tecnologia (REQUIMTE), Departamento de Química, Faculdade de Ciências e Tecnologia, Universidade NOVA de Lisboa, 2829-516 Caparica, Portugal.

Journal of the American Chemical Society
|June 8, 2023
PubMed
まとめ

研究者は光で活性化される超分子トランスポーターを開発し,光スイッチ可能なカリキサレンを使用した. これらのトランスポーターは,細胞膜を介してカチオン性ペプチドの移動を制御し,潜在的光薬学アプリケーションのために光トリガーされた配送を可能にします.

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