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Updated: Jul 11, 2025

Solid Phase Synthesis of a Functionalized Bis-Peptide Using "Safety Catch" Methodology
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サイド・セレクティブ・ソリッド・フェーズ・メタラフォトレドックスNin) - ペプチドのアリレーション

José A C Delgado1,2, Ya-Ming Tian2, Michela Marcon2

  • 1Laboratory for Sustainable Organic Synthesis and Catalysis, Department of Chemistry, Federal University of São Carlos─UFSCar, Rodovia Washington Luís, km 235, SP-310, São Carlos, São Paulo 13565-905, Brazil.

Journal of the American Chemical Society
|November 17, 2023
PubMed
まとめ

この研究は,トリプトファン残基の選択的N-アリレーションを可能にする固相ペプチド合成のための金属光触媒を導入します. 薬の発見のためのペプチド改変能力を拡大します

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