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Updated: Jul 10, 2025

Preparation of N-2-alkoxyvinylsulfonamides from N-tosyl-1,2,3-triazoles and Subsequent Conversion to Substituted Phthalans and Phenethylamines
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Preparation of N-2-alkoxyvinylsulfonamides from N-tosyl-1,2,3-triazoles and Subsequent Conversion to Substituted Phthalans and Phenethylamines

Published on: January 3, 2018

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Rhカルビノイドによるエナンチオセレクティブマルチ機能化

Yu Qian1, Jie Tang1, Xiaoyu Zhou2

  • 1Guangdong Provincial Key Laboratory of Chiral Molecule and Drug Discovery, School of Pharmaceutical Sciences, Sun Yat-sen University, Guangzhou, Guangdong 510006, China.

Journal of the American Chemical Society
|November 22, 2023
PubMed
まとめ

この研究では,ロジウムカルビノイドを用いた最初の非対称三機能化が導入されました. この新しい方法は,単一のステップで3つの新しい結合を形成し,高エナチオ選択性を持つ多様なβ-アミノエステルを効率的に作成します.

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