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Updated: Jul 9, 2025

A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones
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[4 + 1] キャンセル式二重C-H機能化によるN,N-ダイアルキラニリンからのN-アルキリンドールの一般合成

Bowen Zhang1, Frederik R Erb1, Aristidis Vasilopoulos2

  • 1Department of Chemistry, The University of North Carolina at Chapel Hill, Chapel Hill, North Carolina 27599, United States.

Journal of the American Chemical Society
|November 29, 2023
PubMed
まとめ

この研究では,N-アルキリンドール合成のための新しいC-H機能化法が導入されています. N,N-ダイアキラニリンの効率的な二重無効化は,複雑なインドール・スキャファードを作成するための合理化された経路を提供します.

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