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Updated: Jul 5, 2025

Preparation of Enantiopure Non-Activated Aziridines and Synthesis of Biemamide B, D, and epiallo-Isomuscarine
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アトロポセレクティブ・トータル・シンセシス

Longhui Yu1, Yuuya Nagata2, Hugh Nakamura1

  • 1Department of Chemistry, The Hong Kong University of Science and Technology, Clear Water Bay, Hong Kong 999077, China.

Journal of the American Chemical Society
|January 19, 2024
PubMed
まとめ

抗菌剤であるシフナミドBの新合成は,デカグラムスケールSNAr反応とアトロポセレクティブラロックマクロサイクリングを用いて開発された. この方法は,制御されたアトロピソメリスムのユニークなトリプトファン-トリプトファンのクロスリンクを作成します.

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