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Updated: Jul 4, 2025

Construction of Cyclic Cell-Penetrating Peptides for Enhanced Penetration of Biological Barriers
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Published on: September 19, 2022

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形の形状によって駆動される大きなマクロサイクリックペプチドの膜浸透性

Justin H Faris1, Emel Adaligil2, Nataliya Popovych3

  • 1Department of Chemistry and Biochemistry, University of California, Santa Cruz, California 95064, United States.

Journal of the American Chemical Society
|February 8, 2024
PubMed
まとめ

細胞内タンパク質を標的とする重要な課題である 細胞膜の透過性のためにマクロサイクリックペプチドを最適化しました この研究は,難しい標的に対する薬剤発見のためのペプチド図書館の設計を強化します.

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