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Updated: Jun 22, 2025

Measuring G-protein-coupled Receptor Signaling via Radio-labeled GTP Binding
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ナロキソンと協働するμ-オピオイド受容体調節器

Evan S O'Brien1, Vipin Ashok Rangari2, Amal El Daibani2

  • 1Department of Molecular and Cellular Physiology, Stanford University School of Medicine, Stanford, CA, USA.

Nature
|July 3, 2024
PubMed
まとめ

研究者らは,非活性オピオイド受容体 (μOR) を選択的に標的とする新しい化合物を発見した. このネガティブ・アロステリック・モジュレーター (NAM) は,ナロキソンを強化します.

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