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Updated: May 24, 2025

A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones
07:30

A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones

Published on: January 21, 2020

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炭素二重結合に窒素原子を挿入することによって酸化アミネーション

Yannick Brägger1, Ann-Sophie K Paschke1, Nima Nasiri1

  • 1Laboratorium für Organische Chemie, ETH Zürich, Zürich, Switzerland.

Science (New York, N.Y.)
|March 6, 2025
PubMed
まとめ

研究者たちは,炭素と炭素の二重結合に直接窒素を挿入することで,窒素を含む化合物を合成するための新しい方法を開発しました. この多用途な反応は,ハイパーバレンスのヨウ素反応剤を用いて,ニトリル,アミジン,貴重なN-ヘテロサイクルを生成する.

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