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Updated: Sep 10, 2025

Synthesis of Protein Bioconjugates via Cysteine-maleimide Chemistry
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システイン/セレノシステインの生物結合のための後期アロマC-H結合機能化

Zhenguang Zhao1,2, Jian Huang1,3, Yao Cai1

  • 1Institute of Chemistry, The Hebrew University of Jerusalem, Jerusalem 9190401, Israel.

Journal of the American Chemical Society
|August 19, 2025
PubMed
まとめ

研究者達は,ペプチドやタンパク質に 分子を直接結合させるための 銅媒介の方法を開発しました この生物結合技術はシステインとセレノシステインの残留物と 生物互換性のある条件下で作用し,薬の開発における新たな応用が可能である.

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