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Updated: Sep 10, 2025

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BTK阻害剤TL-895との薬物相互作用の責任

Jack C Stromatt1, Eman A Ahmed1, Thomas Drabison1

  • 1The Ohio State University, Columbus, Ohio, United States.

Cancer research communications
|August 22, 2025
PubMed
まとめ

二重のBTK/ BMX阻害剤であるTL-895は,BMXの強力な阻害を示しています. OATP1B1とCYP3A4の基質ですが,薬物相互作用を引き起こす可能性は低いため,組み合わせ療法ではより安全です.

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