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Updated: Sep 10, 2025

A Simple Bioassay for the Evaluation of Vascular Endothelial Growth Factors
09:04

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Published on: March 15, 2016

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VEGFR-2阻害剤としての1,3,4-チアジアゾール誘導体とそのがん治療に対する分子洞察

Pragya Gawande1, Balaji Wamanrao Matore1, Anjali Murmu1

  • 1Laboratory of Drug Discovery and Ecotoxicology, Department of Pharmacy, Guru Ghasidas Vishwavidyalaya (A Central University), Bilaspur, Chhattisgarh, India.

Chemistry & biodiversity
|August 26, 2025
PubMed
まとめ

血管内皮成長因子受容体-2 (VEGFR- 2) を標的にする新しい阻害剤として,がん治療において有望である. これらの化合物は,既存の治療法と比較して,選択性の向上と毒性の低下の可能性を提供します.

キーワード:
1,3,4-チアジアゾール血管新生癌について構造・活動関係 (SAR) とメカニズム血管内皮成長因子受容体-2 (VEGFR-2) 阻害剤

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