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Updated: Sep 10, 2025

A Flow Cytometry-based Assay to Identify Compounds That Disrupt Binding of Fluorescently-labeled CXC Chemokine Ligand 12 to CXC Chemokine Receptor 4
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A Flow Cytometry-based Assay to Identify Compounds That Disrupt Binding of Fluorescently-labeled CXC Chemokine Ligand 12 to CXC Chemokine Receptor 4

Published on: March 10, 2018

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イマチニブ結合に対するカフェインの調節効果: CYP3A4を標的とした分子ドッキング研究

Manuel-Ovidiu Amzoiu1, Georgeta Sofia Popescu2, Emilia Amzoiu1

  • 1Faculty of Pharmacy, University of Medicine and Pharmacy of Craiova, 200638 Craiova, Romania.

Life (Basel, Switzerland)
|August 28, 2025
PubMed
まとめ

カフェインは,イマチニブのCYP3A4酵素への結合に影響することで,その作用を変えることがあります. この相互作用はイマチニブを変化させる可能性があります.

キーワード:
CYP3A4カフェイン併用する薬物相互作用イマチニブ調節効果分子ドッキング

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