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Updated: Sep 9, 2025

A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones
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A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones

Published on: January 21, 2020

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サルフィナートによる4アミノインドールの地域選択C7硫化

Yun Zhang1, Zhehao Zhang2, Yong-Ke He1

  • 1College of Science, Shenyang University of Chemical Technology, Shenyang 110142, China. yk-h@163.com.

Chemical communications (Cambridge, England)
|August 29, 2025
PubMed
まとめ

研究者は,アミノ群のパラディレクション能力を利用して,4-アミノインドールの地域選択C7-H硫化反応を達成した. この方法は,利用可能な硫酸ナイト反応剤を使用して,多様な硫酸ナイトモチーフを効率的に設置します.

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