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Updated: Sep 9, 2025

Preparation of Contiguous Bisaziridines for Regioselective Ring-Opening Reactions
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Preparation of Contiguous Bisaziridines for Regioselective Ring-Opening Reactions

Published on: July 28, 2022

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スピロアジリジンオキシンドールのレジオおよびステレオ特異的な核性C3酸化:エナチオプア3-アジドおよび3-トリアゾール-2-オキシンドールの合成

Ananda Shankar Mondal1,2, Ankita Biswas1,2, Arindam Jana1

  • 1Centre of Biomedical Research, Sanjay Gandhi Post-Graduate Institute of Medical Sciences Campus, Raebareli Road, Lucknow 226014, India.

The Journal of organic chemistry
|August 29, 2025
PubMed
まとめ

新しい方法により,スピロアジリジンオキシンドールの最初の地域およびステレオ特異的アジデーションが可能になり,貴重な3-アジドオキシンドルが得られます. この効率的な合成は,様々なオキシンドール誘導体と薬物結合体の経路を開きます.

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