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Updated: Sep 9, 2025

Efficient Construction of Drug-like Bispirocyclic Scaffolds Via Organocatalytic Cycloadditions of α-Imino γ-Lactones and Alkylidene Pyrazolones
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Efficient Construction of Drug-like Bispirocyclic Scaffolds Via Organocatalytic Cycloadditions of α-Imino γ-Lactones and Alkylidene Pyrazolones

Published on: February 7, 2019

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バイサイクルダイアジリディンの移動反応性を明らかにする:キラルピラゾリンのエナチオセレクティブ合成

Zhili Liu1, Lichao Ning1, Bingqian Yang1

  • 1Key Laboratory of Green Chemistry & Technology, Ministry of Education, College of Chemistry, Sichuan University Chengdu 610064 P. R. China lililin@scu.edu.cn xmfeng@scu.edu.cn.

Chemical science
|August 29, 2025
PubMed
まとめ

この研究は,バイサイクル・ディアジリジンとドナー・アクセプター・サイクロプロパンを含む新しいリング開き/移動カスケード反応を明らかにした. キラル触媒は,高いエナチオ選択性を持つ多様なキラル二水素-1H-ピラゾールを効率的に生成します.

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