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Updated: Sep 9, 2025

A Microwave-Assisted Direct Heteroarylation of Ketones Using Transition Metal Catalysis
07:06

A Microwave-Assisted Direct Heteroarylation of Ketones Using Transition Metal Catalysis

Published on: February 16, 2020

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テトラ置換されたα,β-不飽和ケトンの非対称的水素化:キラル2置換されたサイクロペンチルアリルケトンの利用

Zhengdong Ding1,2, Feng Gao1, Yining Lu1

  • 1Shanghai Key Laboratory for Molecular Engineering of Chiral Drugs, Frontiers Science Center for Transformative Molecules, School of Chemistry and Chemical Engineering, Shanghai Jiao Tong University, 800 Dongchuan Road, Shanghai 200240, China.

Precision chemistry
|August 29, 2025
PubMed
まとめ

研究者らは,テトラ置換アルケンの効率的なイリジウム触媒による非対称な水素化を開発した. この方法は,薬剤にとって重要なキラルケトンを合成し,高収量とステレオ選択性を有します.

キーワード:
2代入サイクロペンチルアリルケトン非対称な水素化キラル・サイクロペンタンイリジウムテトラ置換アルケーン

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