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Updated: Sep 9, 2025

Chemoselective Preparation of 1-Iodoalkynes, 1,2-Diiodoalkenes, and 1,1,2-Triiodoalkenes Based on the Oxidative Iodination of Terminal Alkynes
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Chemoselective Preparation of 1-Iodoalkynes, 1,2-Diiodoalkenes, and 1,1,2-Triiodoalkenes Based on the Oxidative Iodination of Terminal Alkynes

Published on: September 12, 2018

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調節可能なサイト選択性および化学および地域選択性: λ3-ヨウ素媒介のクロス・ヌクレオフィール結合カスケードによって可能となるインドールアルカリド特権性基架の多様化

Zenghui Sun1,2, Ziyi Zhang1, Ran Guo1

  • 1Department of Medicinal Chemistry, School of Pharmacy, Hebei Medical University, 361 East Zhongshan Road, Shijiazhuang 050017, China.

Organic letters
|September 1, 2025
PubMed
まとめ

この研究は,ラムダ3ヨウ素化学を用いた新しい金属のないクロス・ヌクレオフィール結合法を導入している. このアプローチにより,薬剤発見に不可欠な複雑なインドルアルカロイドの合成が可能です.

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