多剤流出ポンプの小分子阻害剤は,外側に開いた形状を結合することによって,抗生物質の活性を強化します

まとめ

研究者らは,NORAの多剤流出ポンプの強力な阻害剤であるIMP-2380を発見しました. この発見はMRSAのようなバクテリアに対する 抗生物質の有効性を高めることで 抗生物質耐性に対抗する新しい戦略を提供します

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