関連する実験動画

Updated: Sep 9, 2025

Facile Preparation of 2Z,4E-Dienamides by the Olefination of Electron-deficient Alkenes with Allyl Acetate
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Facile Preparation of 2Z,4E-Dienamides by the Olefination of Electron-deficient Alkenes with Allyl Acetate

Published on: June 21, 2017

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キューバンのアミド誘導C-Hアセトキシル化

Shota Nagasawa1, Yoshiharu Iwabuchi1

  • 1Graduate School of Pharmaceutical Sciences, Tohoku University, 6-3 Aoba, Aramaki, Aoba-ku, Sendai 980-8578, Japan.

Chemical & pharmaceutical bulletin
|September 3, 2025
PubMed
まとめ

研究者らは,アミド誘導基を用いて,キュバンをアセトキシル化するための新しいパラジウム誘導方法を開発した. この選択的なC-H機能化は強い塩基を回避し,導入されたアセトキシ群の数を制御することができます.

キーワード:
CHの活性化アセトキシル化キューバイソステルパラジウム

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