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Updated: Sep 9, 2025

Efficient Construction of Drug-like Bispirocyclic Scaffolds Via Organocatalytic Cycloadditions of α-Imino γ-Lactones and Alkylidene Pyrazolones
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Efficient Construction of Drug-like Bispirocyclic Scaffolds Via Organocatalytic Cycloadditions of α-Imino γ-Lactones and Alkylidene Pyrazolones

Published on: February 7, 2019

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薬剤化学のためのヘテロスピロサイクルのアプローチ

Carlos Rodríguez-Arias1, Rubén Miguélez1, Yuliia Holota2,3

  • 1Departamento de Química Orgánica e Inorgánica and Instituto Universitario de Química Organometálica "Enrique Moles", Universidad de Oviedo, Julian Clavería 8, 33006 Oviedo, Spain.

Organic letters
|September 5, 2025
PubMed
まとめ

金 ((I) 触媒は,ブロモアルキンから新しいスピロヘテロサイクルを合成することを可能にします. 多様な機能群を備えた この多用途な化合物は 薬の発見において 価値ある構成要素として機能します

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