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Updated: Sep 9, 2025

Synthesis of Antiviral Tetrahydrocarbazole Derivatives by Photochemical and Acid-catalyzed C-H Functionalization via Intermediate Peroxides CHIPS
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Synthesis of Antiviral Tetrahydrocarbazole Derivatives by Photochemical and Acid-catalyzed C-H Functionalization via Intermediate Peroxides CHIPS

Published on: June 20, 2014

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(R) - と (S) - 4 - ハイドロキシ-2- cyclopenten-1-onesの合成: エンテカビール,アバカビール,およびカルボビールの総合合成

Nanlian Li1, Yaopeng Ma1, Chenlong Zhu1

  • 1School of Pharmaceutical Sciences, Nanjing Tech University, 30 South Puzhu Road, Nanjing 211816, China.

The Journal of organic chemistry
|September 5, 2025
PubMed
まとめ

抗ウイルス薬であるエンテカビル,アバカビル,カルボビルのキラルな構成要素は,リパースベースの新合成によって得られます. このグリーン化学のアプローチは,重要な医薬品の工業生産の可能性を秘めています.

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