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Updated: Sep 8, 2025

Efficient Construction of Drug-like Bispirocyclic Scaffolds Via Organocatalytic Cycloadditions of α-Imino γ-Lactones and Alkylidene Pyrazolones
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Efficient Construction of Drug-like Bispirocyclic Scaffolds Via Organocatalytic Cycloadditions of α-Imino γ-Lactones and Alkylidene Pyrazolones

Published on: February 7, 2019

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マニッヒ基からのコンフォーマル・リストリクト・アミノ・サイクロプロパン・フューズド・ラクトン

Mauricio Bahena Garcia1, Victor Fadare1, Zarko Boskovic1

  • 1Department of Medicinal Chemistry, University of Kansas, Lawrence, Kansas 66045, United States.

Organic letters
|September 6, 2025
PubMed
まとめ

マニッヒ基から独特のサイクロプロパン融合ラクトンを生成するための新しい3段階の方法を開発しました. この光化学的アプローチは,潜在的な応用のために,形状的に制限された分子への迅速な経路を提供します.

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