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Updated: Sep 8, 2025

Quantitative Structure-Activity Relationship, Activity Prediction, and Molecular Dynamics of Non-nucleotide Reverse Transcriptase Inhibitors
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多剤耐性調節剤としてのEuphorbia tirucalliのティグリアングリコシド

Lan-Jun Zhang1, Kai-Bo Wang2, Ke-Jing Li3

  • 1State Key Laboratory of Applied Organic Chemistry, College of Chemistry and Chemical Engineering, Lanzhou University, Lanzhou 730000, People's Republic of China; Tea Research Institute, Yunnan Academy of Agricultural Science, Kunming 650201, People's Republic of China.

Bioorganic chemistry
|September 6, 2025
PubMed
まとめ

研究者達は Euphorbia tirucalliから がん細胞の多剤耐性に対抗する新しい化合物を発見しました これらの天然製品はP-グリコプロテインを阻害し,潜在的な新しい治療戦略を提供します.

キーワード:
ディテルペノイドエウフォルビア・ティルカリ多剤耐性調節器チグリアン・グリコシドチルカロシドA-F

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