関連する実験動画

Updated: Feb 16, 2026

A Fluorescence-based Protocol for Preliminary Screening of Protein Synthesis Inhibitors from Natural Sources
10:24

A Fluorescence-based Protocol for Preliminary Screening of Protein Synthesis Inhibitors from Natural Sources

Published on: January 27, 2026

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仮想スクリーニング,合成,インビロアッセイ,分子動力学シミュレーションによる新しいULK1阻害剤の発見

Yifan Yang1, Huijie Han1, Jingjing Li1

  • 1College of Chemistry and Life Science, Beijing University of Technology, Beijing 100124, PR China.

Bioorganic chemistry
|February 14, 2026
PubMed
まとめ

研究者らは,計算的および実験的方法を使用してがん治療のための新しいULK1阻害剤を発見しました. 有望な候補であるD1-D3は,強力なナノモラー活性を示し,新しい抗がん薬の開発のための基盤を提供している.

キーワード:
試験管内測定法 インビトロ測定法分子ダイナミクスシミュレーション有機合成による有機合成です.ULK1 阻害剤 ULK1 阻害剤仮想スクリーニング

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