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Updated: Feb 20, 2026

Preparation of Stable Bicyclic Aziridinium Ions and Their Ring-Opening for the Synthesis of Azaheterocycles
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Preparation of Stable Bicyclic Aziridinium Ions and Their Ring-Opening for the Synthesis of Azaheterocycles

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2H-アジリネからCu触媒制御のTsグループ除去と再挿入経路を通じた多様な置換ピリミジン合成とTosMICsによる2H-アジリネ

Wen Cheng1, Mengfan Li1, Hao Tang1

  • 1School of Perfume and Aroma Technology, Shanghai Institute of Technology, Shanghai 201418, P. R. China. yiwy@sit.edu.cn.

Organic & biomolecular chemistry
|February 18, 2026
PubMed
まとめ

2つの新しい銅触媒反応により,2H-アジリンとTosMICを使用した代用ピリミジンの効率的な合成が可能になりました. これらの方法は,モジュール性を提供し,電子を取り出さない多様な置換物を導入し,合成の可能性を拡大します.

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