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Updated: Aug 18, 2026

Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission
07:16

Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission

Published on: August 16, 2018

エチルβ-カルボリン-3-カルボキシラートは,ベンゾジアゼピン受容体相互作用の差異を示しています

M Nielsen, C Braestrup

    Nature
    |August 7, 1980
    PubMed
    まとめ

    エチルβ-カルボリン-3-カルボキシラート (β-CCE),潜在的内生リガンドは,脳のベンゾジアゼピン受容体と異なる結合をします. これは,ベンゾジアゼピン受容体が均一ではないことを示唆し,潜在的に異なるサブタイプまたは協力性を示す可能性があります.

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