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Updated: Aug 15, 2026

Drug-induced Sensitization of Adenylyl Cyclase: Assay Streamlining and Miniaturization for Small Molecule and siRNA Screening Applications
09:39

Drug-induced Sensitization of Adenylyl Cyclase: Assay Streamlining and Miniaturization for Small Molecule and siRNA Screening Applications

Published on: January 27, 2014

薬理学的ストレスタリウムスシンチグラフィーで,2-サイクロヘキシルメチリデネヒドラジノアデノシン (WRC-0470). 新型,短期間作用のアデノシンA2A受容体アゴニストである

D K Glover1, M Ruiz, J Y Yang

  • 1Department of Medicine, University of Virginia Health Sciences Center, Charlottesville 22908, USA. dkg2w@virginia.edu

Circulation
|October 1, 1996
PubMed
まとめ

新しい選択性アデノシンA2A受容体アゴニストであるWRC-0470は,ストレス画像のために冠動脈を効果的に拡張し,副作用を引き起こすことはありません. これは,薬理学的ストレステストを受ける患者にとってより安全な代替案を提供します.

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