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Updated: Aug 17, 2026

Characterization of G Protein-coupled Receptors by a Fluorescence-based Calcium Mobilization Assay
11:49

Characterization of G Protein-coupled Receptors by a Fluorescence-based Calcium Mobilization Assay

Published on: July 28, 2014

アルファサブユニットのチロシンリン酸化によるGタンパク質Gq/11の活性化

H Umemori1, T Inoue, S Kume

  • 1Department of Oncology, Institute of Medical Science, University of Tokyo, Tokyo 108, Japan.

Science (New York, N.Y.)
|June 20, 1997
PubMed
まとめ

Gq/11タンパク質の受容体活性化には,Galphaq/11サブユニットのチロシンリン酸化が含まれています. このリン酸化は,Gq/11タンパク質の活性化に不可欠であり,受容体相互作用を調節する.

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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators07:41

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

Published on: February 20, 2018

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