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Updated: Jul 18, 2026

Reverse Yeast Two-hybrid System to Identify Mammalian Nuclear Receptor Residues that Interact with Ligands and/or Antagonists
10:51

Reverse Yeast Two-hybrid System to Identify Mammalian Nuclear Receptor Residues that Interact with Ligands and/or Antagonists

Published on: November 15, 2013

アンドロスタンの代謝産物は,CAR-β核受容体と結合し,それを無効化する

B M Forman1, I Tzameli, H S Choi

  • 1The City of Hope National Medical Center, Duarte, California 91010, USA. bforman@gte.net

Nature
|October 23, 1998
PubMed
まとめ

構成的なアンドロスターン受容体-β (CAR-β) の活動は,特定のアンドロスターンステロイドによって抑制されます. これらのステロイドは逆アゴニストとして作用し,CAR-βを逆転させます.

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